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Search Result

Search Results for " dipeptidyl peptidase iv "

Targets

DPP-4

41

Compounds

4

Natural Products

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T11526 DPP-IV-IN-2 H-Lys(4-nitro-Z)-pyrrolidide DPP-4
DPP-IV-IN-2 (H-Lys(4-nitro-Z)-pyrrolidide) is an inhibitor of both DP8/9 and dipeptidyl peptidase IV (IC50s: 0.1 and 0.95 μM).
T1502 Vildagliptin NVP-LAF 237,LAF237 Apoptosis , Ferroptosis , Proteasome , DPP-4
Vildagliptin (LAF237) is a cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Vildagliptin's cyano moiety undergoes hydrolysis and this inactive metabolit...
T36583 Gly-Pro-pNA hydrochloride Gly-Pro p-nitroanilide hydrochloride Proteasome
Gly-Pro-pNA hydrochloride (Gly-Pro p-nitroanilide hydrochloride) is a dipeptidyl peptidase inhibitor that inhibits dipeptidyl peptidase II, dipeptidyl peptidase IV and dipeptidyl peptidase IX.
T78410 Gly-Pro-AMC hydrobromide Gly-Pro-AMC HCl
Gly-Pro-AMC hydrobromide (Gly-Pro-AMC HCl) is a specific fluorescent dye used in cytofluorescence assays to detect Dipeptidyl peptidase IV (DPP-IV) activity.
T67852 Linagliptin Methyldimer Proteasome
Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
T25340 Diprotin A Ile-Pro-Ile DPP-4
Diprotin A (Ile-Pro-Ile) (Ile-Pro-Ile) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.
T78223 γ-Glu-Tyr gamma-Glutamyltyrosine,gamma-GLU-TYR
γ-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide with competitive inhibition of dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.
T68053 Denagliptin GW823093 DPP-4
Denagliptin is a small molecule dipeptidyl peptidase IV (DPP-4) inhibitor for the treatment of endocrine Ü metabolic diseases and can be used in the study of type 2 diabetes.
T21979 P32/98 hemifumarate P32/98 (hemifumarate)(136259-20-6 free base) DPP-4
P32/98 hemifumarate is a dipeptidyl peptidase IV (DPP4) inhibitor with hypoglycemic properties that improves insulin sensitivity and β-cell responsiveness in the Zucker diabetic rat model, and may be useful in studies of...
T8550 NDMC101 Others , NF-κB , Proteasome
NDMC101 is an inhibitor of dipeptidyl peptidase-IV activity in human T cells and exhibits immunomodulatory effects. It also acts as a novel inhibitor of NFATc1 and NF-κB activity.
T27353 Fotagliptin
Fotagliptin is a dipeptidyl peptidase IV inhibitor.
T25341 Diprotin B
Diprotin B is a dipeptidyl peptidase IV inhibitor.
T22886 K 579 Others
K 579 is a dipeptidyl peptidase IV inhibitor.
T70254 FE-999011
FE-999011 is a dipeptidyl peptidase IV inhibitor.
T11049 Diprotin A TFA Ile-Pro-Pro (TFA) Others
Diprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV).
T31378 Denagliptin tosylate GSK-823093,GSK 823093,GW-823093,GW 823093,GSK823093,GW823093
Denagliptin (GW823093 or GSK-823093) is a dipeptidyl peptidase IV (DPP-IV) inhibitor.
T13826 Prodipine hydrochloride Others
Prodipine hydrochloride for purified and plasma Dipeptidyl peptidase IV (DPP IV) from the rabbit (IC50 of 4.5 μM and 30 μM, respectively).
T26941 Camegliptin RO-4876904-001,R1579,RG1579,RO-4876904,R-1579,RG-1579
Cameglipti, a dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type 2 diabetes.
T10082 DPP-IV-IN-1 Others
DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).
T26850 BMS-538305 HCl BMS-538305,BMS538305,BMS 538305,BMS-538305 hydrochloride
BMS-538305 is a potent, selective inhibitor of dipeptidyl peptidase IV (DPP-IV).
T11450 Gosogliptin PF-00734200,PF-734200 Others
Gosogliptin is a potent and selective dipeptidyl peptidase-IV (DPP-IV) inhibitor.
T63698 PK44 phosphate
PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).
T27598 Imigliptin Dihydrochloride Imigliptin
Imigliptin Dihydrochloride, a selective dipeptidyl peptidase IV (DPP-4) inhibitor, is used potentially for the treatment of type II diabetes.
T79911 O-Benzoylhydroxylamine
O-Benzoyl hydroxylamine exhibits properties as a dipeptidyl peptidase-IV (DPP-IV) inhibitor and demonstrates antidiabetic effects[1].
T22747 DPPI 1c hydrochloride Others
DPPI 1c hydrochloride is an inhibitor of dipeptidyl peptidase IV (IC50 = 104 nM) that shows selectivity over enzymes with DPP-like activity (IC50 > 30 μM).
T82178 H-Pro-Pro-Gln-OH
H-Pro-Pro-Gln-OH is an oligopeptide that exhibits potent inhibitory activity against dipeptidyl peptidase-IV (DPP-IV) [1].
T61076 Vildagliptin dihydrate
Vildagliptin dihydrate (LAF237 dihydrate) is a powerful and stable dipeptidyl peptidase IV (DPP-IV) inhibitor, demonstrating selectivity with an IC50 of 3.5 nM in human Caco-2 cells. This compound exhibits exceptional or...
T13069 Talabostat isomer mesylate Others
Talabostat isomer mesylate is an isomer of talabostat mesylate. Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available inhibitor of dipeptidyl peptidase IV (DPP-IV)(Ki of 0.18 nM).
T39481 NVP-DPP728 dihydrochloride NVP-DPP728 dihydrochloride
NVP-DPP728 dihydrochloride is a highly potent, selective, and orally active inhibitor of dipeptidyl peptidase IV (DPP-IV), with a binding affinity (K i ) of 11 nM. This compound proves useful for investigating diabetes m...
T38771 P32/98 P32/98
P32/98 is a potent inhibitor of dipeptidyl peptidase IV . P32/98 improves glucose tolerance, insulin sensitivity and β-cell responsiveness in preclinical studies using the fatty Zucker rat, an animal model for IGT (impai...
T68652 Carmegliptin dihydrochloride
Carmegliptin dihydrochloride is the salt form of Camegliptin (free base), also known as RG-1579 and RO4876904, a dipeptidyl peptidase IV (DPP-4) inhibitor potentially for the treatment of type 2 diabetes.
T68863 MK-0626 free base
MK-0626 is a Dipeptidyl peptidase IV (DPP-4) inhibitor, improving neovascularization by increasing both the number of circulating endothelial progenitor cells and endothelial nitric oxide synthetase expression.
T61414 DPP-4 inhibitor 3
Compound 5a, also known as DPP-4 inhibitor 3, is a powerful dipeptidyl peptidase IV (DPP-IV) inhibitor, demonstrating an IC50 value of 0.75 nM. It exhibits outstanding antioxidant and insulinotropic activity [1].
T63964 DPP-4/GPR119 modulator 2
DPP-4/GPR119 modulator 2 is an inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 0.22 μM) and an agonist of GPR119 (EC50: 0.95 μM).
T68491 Melogliptin
Melogliptin, also known as EMD-675992 and GRC-8200, is a potent and selective a dipeptidyl peptidase IV (DPP-IV) inhibitor potentially for treatment of type II diabetes. Melogliptin significantly reduced HbA1c from b...
T37861 Talabostat
Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM. Talabostat is a nonselective DPP-IV inhibitor, inhibiting DPP8/9, FAP, DPP2 ...
T81025 Teduglutide TFA ALX-0600 TFA
Teduglutide TFA, a dipeptidyl peptidase IV-resistant glucagon-like peptide-2 (GLP-2) analogue, exhibits trophic effects on the gut mucosa and is used in research related to short bowel syndrome (SBS) and Crohn's disease ...
T73875 Fotagliptin benzoate
Fotagliptin benzoate, a Dipeptidyl Peptidase IV (DPP-4) inhibitor with an inhibitory concentration (IC50) of 2.27 nM, demonstrates significant safety in both rat and dog models. It is utilized in Type 2 diabetes mellitus...
T74978 DPP IV/hCA II-IN-1
DPP IV/hCA II-IN-1 is a potent, selective inhibitor of dipeptidyl peptidase IV (DPP IV) and carbonic anhydrase (CA), exhibiting an IC50 of 0.049 μM for DPP IV and K_i values of 0.0361, 0.0428, 0.0941, 0.1328, 0.2615, and...
T21691 NVP DPP 728 dihydrochloride
NVP-DPP728 is a potent, reversible, nitrile-dependent inhibitor of dipeptidyl peptidase IV (DPP-IV), demonstrating an inhibition constant (K i) of 11 nM for human DPP-IV amidolytic activity. By inhibiting the degradation...
T74528 DPP-4/GPR119 modulator 1
DPP-4/GPR119 modulator 1 (Compound 22) is an orally active compound that functions as both a dipeptidyl peptidase IV (DPP-IV) inhibitor and GPR119 agonist. It demonstrates a glucose-lowering effect in blood and exhibits ...

Compounds

DPP-IV-IN-2
T11526
Synonym: H-Lys(4-nitro-Z)-pyrrolidide
Target: DPP-4
Vildagliptin
T1502
Synonym: NVP-LAF 237,LAF237
Target: Apoptosis, Ferroptosis, Proteasome, DPP-4
Gly-Pro-pNA hydrochloride
T36583
Synonym: Gly-Pro p-nitroanilide hydrochloride
Target: Proteasome
Gly-Pro-AMC hydrobromide
T78410
Synonym: Gly-Pro-AMC HCl
Target:
Linagliptin Methyldimer
T67852
Synonym:
Target: Proteasome
Diprotin A
T25340
Synonym: Ile-Pro-Ile
Target: DPP-4
γ-Glu-Tyr
T78223
Synonym: gamma-Glutamyltyrosine,gamma-GLU-TYR
Target:
Denagliptin
T68053
Synonym: GW823093
Target: DPP-4
P32/98 hemifumarate
T21979
Synonym: P32/98 (hemifumarate)(136259-20-6 free base)
Target: DPP-4
NDMC101
T8550
Synonym:
Target: Others, NF-κB, Proteasome
Fotagliptin
T27353
Synonym:
Target:
Diprotin B
T25341
Synonym:
Target:
K 579
T22886
Synonym:
Target: Others
FE-999011
T70254
Synonym:
Target:
Diprotin A TFA
T11049
Synonym: Ile-Pro-Pro (TFA)
Target: Others
Denagliptin tosylate
T31378
Synonym: GSK-823093,GSK 823093,GW-823093,GW 823093,GSK823093,GW823093
Target:
Prodipine hydrochloride
T13826
Synonym:
Target: Others
Camegliptin
T26941
Synonym: RO-4876904-001,R1579,RG1579,RO-4876904,R-1579,RG-1579
Target:
DPP-IV-IN-1
T10082
Synonym:
Target: Others
BMS-538305 HCl
T26850
Synonym: BMS-538305,BMS538305,BMS 538305,BMS-538305 hydrochloride
Target:
Gosogliptin
T11450
Synonym: PF-00734200,PF-734200
Target: Others
PK44 phosphate
T63698
Synonym:
Target:
Imigliptin Dihydrochloride
T27598
Synonym: Imigliptin
Target:
O-Benzoylhydroxylamine
T79911
Synonym:
Target:
DPPI 1c hydrochloride
T22747
Synonym:
Target: Others
H-Pro-Pro-Gln-OH
T82178
Synonym:
Target:
Vildagliptin dihydrate
T61076
Synonym:
Target:
Talabostat isomer mesylate
T13069
Synonym:
Target: Others
NVP-DPP728 dihydrochloride
T39481
Synonym: NVP-DPP728 dihydrochloride
Target:
P32/98
T38771
Synonym: P32/98
Target:
Carmegliptin dihydrochloride
T68652
Synonym:
Target:
MK-0626 free base
T68863
Synonym:
Target:
DPP-4 inhibitor 3
T61414
Synonym:
Target:
DPP-4/GPR119 modulator 2
T63964
Synonym:
Target:
Melogliptin
T68491
Synonym:
Target:
Talabostat
T37861
Synonym:
Target:
Teduglutide TFA
T81025
Synonym: ALX-0600 TFA
Target:
Fotagliptin benzoate
T73875
Synonym:
Target:
DPP IV/hCA II-IN-1
T74978
Synonym:
Target:
NVP DPP 728 dihydrochloride
T21691
Synonym:
Target:
DPP-4/GPR119 modulator 1
T74528
Synonym:
Target:
Cat No. Product Name Synonyms Targets
TN1418 Azaleatin DPP-4
Azaleatin is a natural product from Rhododendron simsii. Azaleatin is a dipeptidyl peptidase-IV inhibitor. Azaleatin can be used for type-2 diabetes and obesity studies.
T16838 Saikogenin A Proteasome , DPP-4
Saikogenin A is a dipeptidyl peptidase-4 inhibitor.
T39219 Ficusonolide
Ficusonolide exhibits significant antidiabetic activity through its interactions with dipeptidyl peptidase-IV (DPP-IV), protein tyrosine phosphatase 1B (PTP-1B), α-glucosidase, and α-amylase.
T81898 Lyciumamide A
DPP-IV-IN-5, derived from Lycium barbarum fruits, demonstrates moderate agonistic activity towards peroxisome proliferator-activated receptor (PPARγ), showing EC50 values between 10.09 and 44.26 μM, and exhibits inhibito...

Natural Products

Azaleatin
TN1418
Synonym:
Target: DPP-4
Saikogenin A
T16838
Synonym:
Target: Proteasome, DPP-4
Ficusonolide
T39219
Synonym:
Target:
Lyciumamide A
T81898
Synonym:
Target:

Recombinant Proteins

Species：
Cynomolgus,Rhesus (1)
Human (1)
Rat (1)
Expression System：
HEK293 Cells (2)
E. coli (1)
Tag：
His (1)
N-6xHis-SUMO (1)
N-His (1)
Cat No. Product Name Species Expression System
TMPH-03279 DPP4/CD26 Protein, Rat, Recombinant (His & SUMO) Rat E. coli
Cell surface glycoprotein receptor involved in the costimulatory signal essential for T-cell receptor (TCR)-mediated T-cell activation. Acts as a positive regulator of T-cell coactivation, by binding at least ADA, CAV1, ...
TMPK-00377 DPPIV/CD26 Protein, Cynomolgus/Rhesus macaque, Recombinant (His) Cynomolgus,Rhesus HEK293 Cells
CD26/dipeptidyl peptidase (DPP)IV is a membrane-bound protein found in many cell types of the body, and a soluble form is present in body fluids. There is longstanding evidence that various primary tumors and also metast...
TMPY-01854 DPP10 Protein, Human, Recombinant (His) Human HEK293 Cells
Inactive dipeptidyl peptidase 1, also known as Dipeptidyl peptidase IV-related protein 3, Dipeptidyl peptidase X, Dipeptidyl peptidase-like protein 2, DPRP-3, DPL2 and DPP1, is a single-pass type II membrane protein w...
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